BDBM712264 (4-Phenylpiperazin-1-yl)(5- (2,4,5-trifluoro-3- hydroxyphenyl)-1,2,4- oxadiazol-3-yl)methanone::US20250011311, Example 81

SMILES O=C(c1noc(-c2cc(F)c(F)c(O)c2F)n1)N1CCN(c2ccccc2)CC1

InChI Key InChIKey=ZSIJWASHWHNGNE-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 712264   

Target17-beta-hydroxysteroid dehydrogenase 13(Human)
Astrazeneca

US Patent
LigandPNGBDBM712264((4-Phenylpiperazin-1-yl)(5- (2,4,5-trifluoro-3- hy...)
Affinity DataIC50: 95nMAssay Description:Final assay conditions were 80 nM of 17bHSD13, 0.5 mM of NAD, 20 μM Estradiol and various concentrations of compound in buffer (5 mM EDTA (TEKNOVA E0...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/22/2025
Entry Details
US Patent