BDBM718131 US20250042862, Compound 92

SMILES N#Cc1ccc(-c2nc(N3CCC(N)CC3)nc3c2CN(c2ccccc2C(F)(F)F)CC3)cc1F

InChI Key InChIKey=PKACXZZOJVBCES-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 718131   

TargetLysine-specific histone demethylase 1A(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM718131(US20250042862, Compound 92)
Affinity DataIC50: 165nMAssay Description:The purpose of this experiment was to test the in vitro inhibitory activity of the compounds against LSD1. The human recombinant LSD1 protein used in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/12/2025
Entry Details
US Patent