BDBM720168 6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazol-4-yl]methoxy}-2-(oxolan-3-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine::US20250051323, Example 9

SMILES Cc1ccc(-c2noc(C)c2COc2cc3c(cn2)CN(C2CCOC2)CC3)cn1

InChI Key InChIKey=BEEKOIOWKJWHPN-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 720168   

TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
Richter Gedeon

US Patent
LigandPNGBDBM720168(6-{[5-methyl-3-(6-methylpyridin-3-yl)-1,2-oxazol-4...)
Affinity DataKi:  4.90nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampule of membrane homogenate was thawed and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
US Patent