BDBM720178 3-{[3-({5-methyl-3-[6-(trifluoromethyl)pyridin-3-yl}-1,2-oxazol-4-yl]methoxy)-5H,6H,7H,8H-pyrido[3,4-c]pyridazin-7-yl]methyl}-1lambda6-thiolane-1,1-dione tartarate salt::US20250051323, Example 19

SMILES Cc1onc(-c2ccc(C(F)(F)F)nc2)c1COc1cc2c(nn1)CN(CC1CCS(=O)(=O)C1)CC2

InChI Key InChIKey=PSKPLVJLHZSRKF-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 720178   

TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Human)
Richter Gedeon

US Patent
LigandPNGBDBM720178(3-{[3-({5-methyl-3-[6-(trifluoromethyl)pyridin-3-y...)
Affinity DataKi:  35.5nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampule of membrane homogenate was thawed and...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/17/2025
Entry Details
US Patent