BDBM727059 US12252493, Example 11

SMILES Cc1cc(C2=CN=C(NCc3c(F)ccc4c3CCO4)N3CC([C@@H](C)N)N=C23)n(C)n1

InChI Key InChIKey=XKMMCRANAIDZBC-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 727059   

LigandPNGBDBM727059(US12252493, Example 11)
Affinity DataIC50: 375nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
7/22/2025
Entry Details
US Patent