BDBM727093 US12252493, Example 43

SMILES Cc1cc(-c2cnc(NCc3c(F)ccc4c3CCO4)n3cc(-c4nn[nH]n4)nc23)n(C)n1

InChI Key InChIKey=ARVNNNAHZHBLFN-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 727093   

TargetHistone-binding protein RBBP4/Histone-lysine N-methyltransferase EZH2/Polycomb protein EED/Polycomb protein SUZ12/Zinc finger protein AEBP2(Human)
Mirati Therapeutics

US Patent

LigandBDBM727093(US12252493, Example 43)Copy SMILESCopy InChI

Affinity DataIC50: 250nMAssay Description:Briefly, compounds of the present invention were solubilized in DMSO and a series of 10, three-fold serial dilutions were made for each compound in 1...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
7/22/2025
Entry Details
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