BDBM728162 (Z)-1-acetyl-2-((4- (2-acetyl-1,2,3,4- tetrahydroisoquin- olin-7-yl)-6- (((tetrahydro-2H- pyran-4-yl)amino)- methyl)quinolin- 2-yl)methylene)- indolin-3-one::US20250091994, Example 211
SMILES CC(=O)N1CCc2ccc(-c3cc(/C=C4/C(=O)c5ccccc5N4C(C)=O)nc4ccc(CNC5CCOCC5)cc34)cc2C1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 728162
TargetRAF proto-oncogene serine/threonine-protein kinase [50-131]/GTPase KRas [G12V](Human)
Kobe University
US Patent
Kobe University
US Patent
Affinity DataIC50: 600nMAssay Description:The in vitro Ras-Raf binding inhibitory activity of the compound of the present invention was evaluated by an ELISA method described below. GST-c-Raf...More data for this Ligand-Target Pair
