BDBM730780 US20250122182, Syn. Ex. 101

SMILES CCc1ccc(OCCNC(=O)OCC2c3ccccc3C3C=CC=CC32)c(S(=O)(=O)Nc2noc3cc(Cn4cc(CNC(=O)OC)cn4)cc(OC)c23)c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 730780   

TargetHistone acetyltransferase KAT6A(Human)
Isosterix

US Patent
LigandPNGBDBM730780(US20250122182, Syn. Ex. 101)
Affinity DataIC50: 4nMAssay Description:The Kat6a inhibitory activity of test compounds was determined using an Alpha Screen-based detection method. The assay reactions were conducted in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetHistone acetyltransferase KAT6B(Human)
Isosterix

US Patent
LigandPNGBDBM730780(US20250122182, Syn. Ex. 101)
Affinity DataIC50: 2.49E+3nMAssay Description:The Kat6a inhibitory activity of test compounds was determined using an Alpha Screen-based detection method. The assay reactions were conducted in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent