BDBM730786 US20250122182, Syn. Ex. 50

SMILES COC(=O)NCc1cnn(Cc2cc(OC(F)F)c3c(NS(=O)(=O)c4c(OC)cccc4OC)noc3c2)c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 730786   

TargetHistone acetyltransferase KAT6A(Human)
Isosterix

US Patent
LigandPNGBDBM730786(US20250122182, Syn. Ex. 50)
Affinity DataIC50: 34nMAssay Description:The Kat6a inhibitory activity of test compounds was determined using an Alpha Screen-based detection method. The assay reactions were conducted in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent

TargetHistone acetyltransferase KAT6B(Human)
Isosterix

US Patent
LigandPNGBDBM730786(US20250122182, Syn. Ex. 50)
Affinity DataIC50: 2.40E+3nMAssay Description:The Kat6a inhibitory activity of test compounds was determined using an Alpha Screen-based detection method. The assay reactions were conducted in a ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/18/2025
Entry Details
US Patent