BDBM731939 3-fluoro-N-[2-[3- (fluoromethyl)azetidin-1- yl]ethyl]-4-[(1R,3R)-2-(2- fluoro-2-methyl-propyl)-3- methyl-1,3,4,9- tetrahydropyrido[3,4-b]indol- 1-yl]aniline::US20250114338, Example 322

SMILES C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2ccc(NCCN3CC(CF)C3)cc2F)N1CC(C)(C)F

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 731939   

TargetEstrogen receptor(Human)
Genentech

US Patent
LigandPNGBDBM731939(3-fluoro-N-[2-[3- (fluoromethyl)azetidin-1- yl]eth...)
Affinity DataEC50:  0.0250nMAssay Description:All of the exemplary Formula I compounds in Tables 1 and 2 were tested for binding to ERa (Estrogen Receptor alpha) and biological activity according...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
8/22/2025
Entry Details
US Patent