BDBM732083 (R)-3-((1R,3R)-1-(2,6- difluoro-4-(2-(3- (fluoromethyl)azetidin-1- yl)ethoxy)phenyl)-3-methyl- 3,4-dihydro-1H-pyrido[3,4- b]indol-2(9H)-yl)-2- (fluoromethyl)propan-1-ol::US20250114338, Example 402

SMILES C[C@@H]1Cc2c([nH]c3ccccc23)[C@@H](c2c(F)cc(OCCN3CC(CF)C3)cc2F)N1C[C@H](CO)CF

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 732083   

TargetEstrogen receptor(Human)
Genentech

US Patent
LigandPNGBDBM732083((R)-3-((1R,3R)-1-(2,6- difluoro-4-(2-(3- (fluorome...)
Affinity DataEC50:  0.0320nMAssay Description:All of the exemplary Formula I compounds in Tables 1 and 2 were tested for binding to ERa (Estrogen Receptor alpha) and biological activity according...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
8/22/2025
Entry Details
US Patent