BDBM734332 1-[(3R)-2,2-Dimethyl-3-{[6-methyl-5-(1-methyl-1H-imidazol-4-yl)pyridin-2-yl]amino}pyrrolidin-1-yl]-2-(4-fluorophenyl)ethan-1-one (3A) and 1-[(3S)-2,2-Dimethyl-3-{[6-methyl-5-(1-methyl-1H-imidazol-4-yl)pyridin-2-yl]amino}pyrrolidin-1-yl]-2-(4-fluorophenyl)ethan-1-one (3B)::US20250129048, Example 3B

SMILES Cc1nc(N[C@@H]2CCN(C(=O)OC(C)(C)C)C2(C)C)ccc1-c1cn(C)cn1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 734332   

TargetMelanocortin receptor 4(Human)
Pfizer

US Patent
LigandPNGBDBM734332(1-[(3R)-2,2-Dimethyl-3-{[6-methyl-5-(1-methyl-1H-i...)
Affinity DataKi:  4.20nMAssay Description:The binding affinity of test compounds at the α-melanocyte-stimulating hormone receptor (hMC4R) was assessed using a radioligand competition binding ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
8/25/2025
Entry Details
US Patent