BDBM734445 US20250129068, Example 8

SMILES COc1ncccc1S(=O)(=O)Nc1nccc(C#Cc2cnc3[nH]ncc3c2)c1F

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 734445   

TargeteIF-2-alpha kinase GCN2(Human)
IP2IPO Innovations

US Patent
LigandPNGBDBM734445(US20250129068, Example 8)
Affinity DataKi:  59.9nMAssay Description:The inhibitory activity of the Example compounds towards GCN2 enzyme was measured according to the description below, using a LanthaScreen TR-FRET (T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
8/25/2025
Entry Details
US Patent