BDBM736475 N-((2,6-dimethoxyphenyl)sulfonyl)- 3-methoxy-4-((thiazol-2- yloxy)methyl)benzamide::US20250136553, Compound 58

SMILES COc1cc(C(=O)NS(=O)(=O)c2c(OC)cccc2OC)ccc1COc1nccs1

InChI Key InChIKey=HNYKMFCURHBEJS-UHFFFAOYSA-N

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736475   

TargetHistone acetyltransferase KAT6A(Human)
Olema Pharmaceuticals

US Patent
LigandChemical structure of BindingDB Monomer ID 736475BDBM736475(N-((2,6-dimethoxyphenyl)sulfonyl)- 3-methoxy-4-((t...)
Affinity DataIC50: 177nMAssay Description:TR-FRET based methods were used for assaying compounds of the present invention for KAT6A enzyme inhibitory activity. TR-FRET is a homogeneous proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/2/2025
Entry Details
US Patent