BDBM736508 5-((1H-pyrazol-1-yl)methyl)-N-((2-(difluoromethoxy)-6- methoxyphenyl)sulfonyl)-6-methoxypicolinamide::US20250136553, Compound 220

SMILES COc1cccc(OC(F)F)c1S(=O)(=O)NC(=O)c1ccc(Cn2cccn2)c(OC)n1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736508   

LigandPNGBDBM736508(5-((1H-pyrazol-1-yl)methyl)-N-((2-(difluoromethoxy...)
Affinity DataIC50: 7nMAssay Description:TR-FRET based methods were used for assaying compounds of the present invention for KAT6A enzyme inhibitory activity. TR-FRET is a homogeneous proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TBA
Entry Details
US Patent