BDBM736545 5-((1H-pyrazol-1-yl)methyl)-6-methoxy-N-((2,4,6- tris(methoxy-d3)phenyl)sulfonyl)picolinamide::US20250136553, Compound 270

SMILES [2H]C([2H])([2H])Oc1cc(OC([2H])([2H])[2H])c(S(=O)(=O)NC(=O)c2ccc(Cn3cccn3)c(OC)n2)c(OC([2H])([2H])[2H])c1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736545   

LigandPNGBDBM736545(5-((1H-pyrazol-1-yl)methyl)-6-methoxy-N-((2,4,6- t...)
Affinity DataIC50: 6nMAssay Description:TR-FRET based methods were used for assaying compounds of the present invention for KAT6A enzyme inhibitory activity. TR-FRET is a homogeneous proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
TBA
Entry Details
US Patent