BDBM736554 5-((1H-pyrazol-1-yl)methyl)-N-((5-(tert-butyl)-2,3- dihydrobenzofuran-7-yl)sulfonyl)-6-methoxypicolinamide::US20250136553, Compound 280

SMILES COc1nc(C(=O)NS(=O)(=O)c2cc(C(C)(C)C)cc3c2OCC3)ccc1Cn1cccn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 736554   

LigandPNGBDBM736554(5-((1H-pyrazol-1-yl)methyl)-N-((5-(tert-butyl)-2,3...)
Affinity DataIC50: 5nMAssay Description:TR-FRET based methods were used for assaying compounds of the present invention for KAT6A enzyme inhibitory activity. TR-FRET is a homogeneous proxim...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
TBA
Entry Details
US Patent