BDBM739767 (S)-1-(3-(4-amino-7-(cyclopropanecarbonyl)-3-((2-methyl-2H-indazol-6-yl)ethynyl)-1H-pyrazolo[4,3-c]pyridin-1-yl)pyrrolidin-1-yl)prop-2-en-1-one::US20250152564, Example 84

SMILES C=CC(=O)N1CC[C@H](n2nc(C#Cc3ccc4cn(C)nc4c3)c3c(N)ncc(C(=O)C4CC4)c32)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 739767   

LigandPNGBDBM739767((S)-1-(3-(4-amino-7-(cyclopropanecarbonyl)-3-((2-m...)
Affinity DataIC50: 0.300nMAssay Description:TR-FRET (time-resolved fluorescence resonance energy transfer) method was used to detect the inhibitory activity of the compounds on FGFR1, FGFR2, FG...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM739767((S)-1-(3-(4-amino-7-(cyclopropanecarbonyl)-3-((2-m...)
Affinity DataIC50: 0.5nMAssay Description:TR-FRET (time-resolved fluorescence resonance energy transfer) method was used to detect the inhibitory activity of the compounds on FGFR1, FGFR2, FG...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM739767((S)-1-(3-(4-amino-7-(cyclopropanecarbonyl)-3-((2-m...)
Affinity DataIC50: 1nMAssay Description:TR-FRET (time-resolved fluorescence resonance energy transfer) method was used to detect the inhibitory activity of the compounds on FGFR1, FGFR2, FG...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent