BDBM744008 N-(5-((4-Ethylpiperazin-1-yl)methyl) pyridin-2-yl)-1-isopropyl-1H-[1,2,3]tri- azolo[4,5-h]quinazolin-8-amine hydrochloride::US12312355, Compound I-10

SMILES CCN1CCN(Cc2ccc(Nc3ncc4ccc5nnn(C(C)C)c5c4n3)nc2)CC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 744008   

LigandPNGBDBM744008(N-(5-((4-Ethylpiperazin-1-yl)methyl) pyridin-2-yl)...)
Affinity DataIC50: 10nMAssay Description:The inhibitory effect of the compound on the kinase CDK4/cyclin D3 was tested by the Caliper Mobility Shift Assay method. The final test concentratio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM744008(N-(5-((4-Ethylpiperazin-1-yl)methyl) pyridin-2-yl)...)
Affinity DataIC50: 30nMAssay Description:The inhibitory effect of the compound on the kinase CDK4/cyclin D3 was tested by the Caliper Mobility Shift Assay method. The final test concentratio...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent