BDBM746828 (E)-N-(3-fluoro-2-methylphenyl)-3-(1-methyl-2-oxo-2,3-dihydro-1H-benzo[d]imidazol-5-yl)acrylamide::US20250179028, Example 7

SMILES Cc1c(F)cccc1NC(=O)/C=C/c1ccc2c(c1)[nH]c(=O)n2C

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 746828   

TargetCytochrome P450 2D6(Human)
NRG Therapeutics

US Patent
LigandPNGBDBM746828((E)-N-(3-fluoro-2-methylphenyl)-3-(1-methyl-2-oxo-...)
Affinity DataIC50: 3.00E+4nMAssay Description:Studies to assess tested compound mediated inhibition of cytochrome P450 enzyme isoform CYP2D6 were performed using human liver microsomes (BD Gentes...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/30/2025
Entry Details
US Patent