BDBM748856 2-pyrazolo[1,5-a]pyridin-2-yl-N-[4-[3-(2-pyridyl)-1H-pyrrolo[3,2-b]pyridin-2-yl]-2-pyridyl]acetamide::US20250188075, Example 15

SMILES O=C(Cc1cc2ccccn2n1)Nc1cc(-c2[nH]c3cccnc3c2-c2ccccn2)ccn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 748856   

LigandPNGBDBM748856(2-pyrazolo[1,5-a]pyridin-2-yl-N-[4-[3-(2-pyridyl)-...)
Affinity DataIC50: 1.07nMAssay Description:For the assay 50 nl of a 100-fold concentrated solution of the test compound in DMSO was pipetted into a white 1536-well microtiter plate (Greiner Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM748856(2-pyrazolo[1,5-a]pyridin-2-yl-N-[4-[3-(2-pyridyl)-...)
Affinity DataIC50: 3.75nMAssay Description:For the assay 50 nl of a 100-fold concentrated solution of the test compound in DMSO was pipetted into a white 1536-well microtiter plate (Greiner Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM748856(2-pyrazolo[1,5-a]pyridin-2-yl-N-[4-[3-(2-pyridyl)-...)
Affinity DataIC50: 10.3nMAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a white 1536-well microtiter plate (Greiner Bi...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM748856(2-pyrazolo[1,5-a]pyridin-2-yl-N-[4-[3-(2-pyridyl)-...)
Affinity DataIC50: 24.2nMAssay Description:For the assay 50 nl of a 100 fold concentrated solution of the test compound in DMSO was pipetted into a white low volume 384-well microtiter plate (...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent