BDBM754288 Ethyl ((3-((2-(difluoromethoxy)-6-methylpyridin-3-yl)carbamoyl)-3-(2-isopropylphenyl)azetidin-1-yl)sulfonyl)glycinate::US12344597, Example 15-1

SMILES CCOC(=O)CNS(=O)(=O)N1CC(C(=O)Nc2ccc(C)nc2OC(F)F)(c2ccccc2C(C)C)C1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 754288   

TargetLysophosphatidic acid receptor 1(Human)
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM754288(Ethyl ((3-((2-(difluoromethoxy)-6-methylpyridin-3-...)
Affinity DataIC50: 5nMAssay Description:The Tango™ EDG2-bla U2OS cells are obtained from Invitrogen. These cells contain the human LPA1 receptor cDNA linked to a TEV protease site and a Gal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent