BDBM754354 1-(N-(N-acetylsulfamoyl)-N-methylglycyl)-N-(2-(difluoromethoxy)-6-methylpyridin-3-yl)-3-(2-isopropylphenyl)azetidine-3-carboxamide::US12344597, Example 16-5

SMILES CC(=O)NS(=O)(=O)N(C)CC(=O)N1CC(C(=O)Nc2ccc(C)nc2OC(F)F)(c2ccccc2C(C)C)C1

InChI Key InChIKey=DPOSAKDDGGXCMB-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 754354   

TargetLysophosphatidic acid receptor 1(Human)
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM754354(1-(N-(N-acetylsulfamoyl)-N-methylglycyl)-N-(2-(dif...)
Affinity DataIC50: 47nMAssay Description:The Tango™ EDG2-bla U2OS cells are obtained from Invitrogen. These cells contain the human LPA1 receptor cDNA linked to a TEV protease site and a Gal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
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