BDBM754417 2-(4-((2-(difluoromethoxy)-6-methylpyridin-3-yl)carbamoyl)-4-(2-isopropylphenyl)piperidine-1-carboxamido)ethyl methacrylate::US12344597, Example 17-21

SMILES C=C(C)C(=O)OCCNC(=O)N1CCC(C(=O)Nc2ccc(C)nc2OC(F)F)(c2ccccc2C(C)C)CC1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 754417   

TargetLysophosphatidic acid receptor 1(Human)
Idorsia Pharmaceuticals

US Patent
LigandPNGBDBM754417(2-(4-((2-(difluoromethoxy)-6-methylpyridin-3-yl)ca...)
Affinity DataIC50: 5nMAssay Description:The Tango™ EDG2-bla U2OS cells are obtained from Invitrogen. These cells contain the human LPA1 receptor cDNA linked to a TEV protease site and a Gal...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/22/2025
Entry Details
US Patent