BDBM755819 US20250214986, Compound of formula I

SMILES Cc1cnc(-c2cc(O[C@@H](C)[C@@H](C)O)cc(C(=O)N[C@H](C)c3cnc(C(F)(F)F)nc3)c2F)s1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 755819   

TargetP2X purinoceptor 3(Human)
Humanwell Heathcare (Group)

US Patent
LigandPNGBDBM755819(US20250214986, Compound of formula I)
Affinity DataIC50: 67nMAssay Description:The antagonistic activity of human P2X3 receptor (hP2X3) antagonists against hP2X3 was evaluated using the FLIPR Calcium 4 Assay Kit (Molecular Devic...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent