BDBM755983 3-(5-(7-(azetidin-1-ylmethyl)-1- ethyl-1H-pyrrolo[3,2-b]pyridin-5- yl)-1-oxoisoindolin-2- yl)piperidine-2,6-dione::US20250214991, Compound 124

SMILES CCn1ccc2nc(-c3ccc4c(c3)CN(C3CCC(=O)NC3=O)C4=O)cc(CN3CCC3)c21

InChI Key InChIKey=MPMGBJYXRHTGTN-UHFFFAOYSA-N

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 755983   

TargetDNA damage-binding protein 1/Protein cereblon(Human)
Oncopia Therapeutics, Inc. D/B/A/ Sk Life Science Labs

US Patent
LigandChemical structure of BindingDB Monomer ID 755983BDBM755983(3-(5-(7-(azetidin-1-ylmethyl)-1- ethyl-1H-pyrrolo[...)
Affinity DataIC50: 5.00E+3nMAssay Description:The binding potency was determined using HTRF assay technology (Perkin Elmer). Compounds were serially diluted in DMSO and 0.2 μL volume was transfer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/23/2025
Entry Details
US Patent