BDBM756402 2-(((2S)-4-(2-(4-chlorophenyl)-2,3-dihydrobenzo[b][1,4]dioxin-5-yl)-2-methylpiperazin-1-yl)methyl)-3-(((S)-oxetan-2-yl)methyl)-3H-imidazo[4,5-b]pyridine-5-carboxylic acid ::US20250214999, Compound 114a

SMILES C[C@H]1CN(c2cccc3c2OCC(c2ccc(Cl)cc2)O3)CCN1Cc1nc2ccc(C(=O)O)nc2n1C[C@@H]1CCO1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 756402   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM756402(2-(((2S)-4-(2-(4-chlorophenyl)-2,3-dihydrobenzo[b]...)
Affinity DataEC50:  10.1nMAssay Description:Activation of GLP-1 receptor is known to stimulate cyclic AMP (cAMP) production in cells which indicates primary coupling to the Gαs subunit of the G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/24/2025
Entry Details
US Patent