BDBM756415 2-((4-(2-(4-chloro-2-fluorophenyl) chroman-5-yl)piperazin-1-yl)methyl)-3-((S)oxetan-2-ylmethyl)-3H-imidazo[4,5-b]pyridine-5-carboxylic acid ::US20250214999, Compound 123a

SMILES O=C(O)c1ccc2nc(CN3CCN(c4cccc5c4CCC(c4ccc(Cl)cc4F)O5)CC3)n(C[C@@H]3CCO3)c2n1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 756415   

TargetGlucagon-like peptide 1 receptor(Human)
Gasherbrum Bio

US Patent
LigandPNGBDBM756415(2-((4-(2-(4-chloro-2-fluorophenyl) chroman-5-yl)pi...)
Affinity DataEC50:  110nMAssay Description:Activation of GLP-1 receptor is known to stimulate cyclic AMP (cAMP) production in cells which indicates primary coupling to the Gαs subunit of the G...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/24/2025
Entry Details
US Patent