BDBM756777 US20250215014, Compound 119::US20250223301, Compound 119

SMILES CC[C@H]1CN([C@@H](CC)c2nc(C3CC3)no2)[C@H](CC)CN1c1nc2nncn2c2ccc(C#N)nc12

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 756777   

TargetDiacylglycerol kinase alpha(Human)
Inventisbio

US Patent
LigandPNGBDBM756777(US20250215014, Compound 119 | US20250223301, Compo...)
Affinity DataIC50: 3nMAssay Description:The DGKa and DGKz kinase assays were performed using Promega ADP-Glo kit (Promega, Cat #V9102). One microliter test compound was added to a 384-well ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/27/2025
Entry Details
US Patent

TargetDiacylglycerol kinase zeta(Human)
Inventisbio

US Patent
LigandPNGBDBM756777(US20250215014, Compound 119 | US20250223301, Compo...)
Affinity DataIC50: 10nMAssay Description:The DGKa and DGKz kinase assays were performed using Promega ADP-Glo kit (Promega, Cat #V9102). One microliter test compound was added to a 384-well ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/26/2025
Entry Details
US Patent

TargetDiacylglycerol kinase alpha(Human)
Inventisbio

US Patent
LigandPNGBDBM756777(US20250215014, Compound 119 | US20250223301, Compo...)
Affinity DataIC50: 10nMAssay Description:The DGKa and DGKz kinase assays were performed using Promega ADP-Glo kit (Promega, Cat #V9102). One microliter test compound was added to a 384-well ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/26/2025
Entry Details
US Patent

TargetDiacylglycerol kinase zeta(Human)
Inventisbio

US Patent
LigandPNGBDBM756777(US20250215014, Compound 119 | US20250223301, Compo...)
Affinity DataIC50: 21nMAssay Description:The DGKa and DGKz kinase assays were performed using Promega ADP-Glo kit (Promega, Cat #V9102). One microliter test compound was added to a 384-well ...More data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/27/2025
Entry Details
US Patent