BDBM757465 US12357603, Example 103

SMILES COc1cc(S(=O)(=O)NC(=O)c2cc3ccc(N(C)C)cc3o2)cc(Cn2cccn2)c1OC

InChI Key InChIKey=ITXCNPNLLOCRJE-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 757465   

TargetHistone Acetyltransferase KAT6A [194-810]/Zinc Finger Protein Neuro-d4 (DPF1)/ Histone Acetyltransferase Type B Catalytic Subunit (HAT1)(Homo sapiens (Human))
Bayer Aktiengesellschaft

US Patent

LigandBDBM757465(US12357603, Example 103)Copy SMILESCopy InChI

Affinity DataIC50: 1.21E+3nMAssay Description:Recombinant human His-tagged Kat6a protein (amino acids 194-810), was purified in-house from Baculovirus-infected insect cells (Sf9). Histone H4 pept...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
10/28/2025
Entry Details
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