BDBM757568 5-Bromo-N-[2-(cyclopropyloxy)benzene-1-sulfonyl]-6-(dimethylamino)-1-benzofuran-2-carboxamide::US12357603, Example 207

SMILES CN(C)c1cc2oc(C(=O)NS(=O)(=O)c3ccccc3OC3CC3)cc2cc1Br

InChI Key InChIKey=VBDCFMUHZCOUJB-UHFFFAOYSA-N

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 757568   

TargetHistone Acetyltransferase KAT6A [194-810]/Zinc Finger Protein Neuro-d4 (DPF1)/ Histone Acetyltransferase Type B Catalytic Subunit (HAT1)(Homo sapiens (Human))
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US Patent

LigandBDBM757568(5-Bromo-N-[2-(cyclopropyloxy)benzene-1-sulfonyl]-6...)Copy SMILESCopy InChI

Affinity DataIC50: 6.81E+3nMAssay Description:Recombinant human His-tagged Kat6a protein (amino acids 194-810), was purified in-house from Baculovirus-infected insect cells (Sf9). Histone H4 pept...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sid

In Depth
Date in BDB:
10/28/2025
Entry Details
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