BDBM758664 (Racemic) 2''-chloro-N-(6-((4- hydroxyphenyl)amino)-4,5,6,7- tetrahydrobenzo[d]thiazol-2-yl)-5''- methoxy-6-methyl-[4,4''-bipyridine]-3- carboxamide::US20250230171, Compound 135

SMILES COc1cnc(Cl)cc1-c1cc(C)ncc1C(=O)Nc1nc2c(s1)CC(Nc1ccc(O)cc1)CC2

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 758664   

TargetDNA polymerase theta (POLQ) (2-894)(Human)
Moma Therapeutics

US Patent
LigandPNGBDBM758664((Racemic) 2'-chloro-N-(6-((4- hydroxyphenyl)amino)...)
Affinity DataIC50: 8nMAssay Description:POLθ-mediated ATP hydrolysis was measured using the ADP-Glo Kinase Assay (Promega Corporation, Madison, WI). Reactions were performed in white 384-we...More data for this Ligand-Target Pair
Target InfoPDB
GoogleScholar
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/30/2025
Entry Details
US Patent