BDBM759976 US20250236609, Example 85
SMILES Cc1cnc(NC(=O)C2CC2)cc1-c1cc(N2CCN(S(=O)(=O)CC3CC3)C[C@@H]2C)[nH]c(=O)c1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 759976
TargetPhosphatidylinositol 3-kinase catalytic subunit type 3(Human)
Deciphera Pharmaceuticals
US Patent
Deciphera Pharmaceuticals
US Patent
Affinity DataIC50: 100nMAssay Description:Activity of VPS34 kinase was determined using an ADP-Glo kinase activity assay (Promega Corp). Assays were conducted in 384-well plates (5 μL assay v...More data for this Ligand-Target Pair
