BDBM760333 1-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- yl]methoxy}-5H,6H,7H- pyrrolo[3,4-b]pyridin-6-yl)-2- methanesulfonylethan-1- one::US12370182, Example 49

SMILES Cc1onc(-c2ccc(F)cc2)c1COc1ccc2c(n1)CN(C(=O)CS(C)(=O)=O)C2

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 760333   

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandPNGBDBM760333(1-(2-{[3-(4-fluorophenyl)-5- methyl-1,2-oxazol-4- ...)
Affinity DataKi:  1.20nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
11/10/2025
Entry Details
US Patent