BDBM760353 1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triazol-5- yl]methoxy}-5,7-dihydro-6H- pyrrolo[3,4-b]pyridin-6- yl)propan-1-one::US12370182, Example 69

SMILES CCC(=O)N1Cc2ccc(OCc3c(-c4ccc(F)cc4)nnn3C)nc2C1

InChI Key

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 760353   

TargetGamma-aminobutyric acid receptor subunit alpha-5(Human)
Richter Gedeon

US Patent
LigandPNGBDBM760353(1-(2-{[4-(4-fluorophenyl)-1- methyl-1H-1,2,3-triaz...)
Affinity DataKi:  25nMAssay Description:Receptor binding assays were performed in 96-well format in deep-well plates. For each 96-well plate one ampulle of membrane homogenate was thawed an...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
11/10/2025
Entry Details
US Patent