BDBM760851 (3R)-4-[7-(6-Methanesulfonyl-2-methylpyridin-3-yl)-3-(3-methyl-1H-pyrazol-5-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]-3-methylmorpholine ::US12371430, Compound 13
SMILES Cc1cc(-c2n[nH]c3c(-c4ccc(S(C)(=O)=O)nc4C)cc(N4CCOC[C@H]4C)nc23)[nH]n1
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 760851
Affinity DataIC50: 1.40nMAssay Description:The ATR/ATRIP enzymatic assay is performed as a TR-FRET-(HTRF™, Cisbio Bioassays) based 384-well assay. In a first step, purified human recombinant A...More data for this Ligand-Target Pair
