BDBM760879 (3R)-4-[7-(4-Methanesulfonylphenyl)-1-(propan-2-yl)-3-(1H-pyrazol-3-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]-3-methylmorpholine ::US12371430, Compound 41

SMILES CC(C)n1nc(-c2cc[nH]n2)c2nc(N3CCOC[C@H]3C)cc(-c3ccc(S(C)(=O)=O)cc3)c21

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 760879   

LigandPNGBDBM760879((3R)-4-[7-(4-Methanesulfonylphenyl)-1-(propan-2-yl...)
Affinity DataIC50: 1.30nMAssay Description:The ATR/ATRIP enzymatic assay is performed as a TR-FRET-(HTRF™, Cisbio Bioassays) based 384-well assay. In a first step, purified human recombinant A...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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Date in BDB:
TBA
Entry Details
US Patent