BDBM760916 (3R)-3-Methyl-4-[1-methyl-7-(4-methylpyrimidin-5-yl)-3-(1H-pyrazol-3-yl)-1H-pyrazolo[4,3-b]pyridin-5-yl]morpholine ::US12371430, Compound 87
SMILES Cc1ncncc1-c1cc(N2CCOC[C@H]2C)nc2c(-c3cc[nH]n3)nn(C)c12
InChI Key
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 760916
Affinity DataIC50: 0.400nMAssay Description:The ATR/ATRIP enzymatic assay is performed as a TR-FRET-(HTRF™, Cisbio Bioassays) based 384-well assay. In a first step, purified human recombinant A...More data for this Ligand-Target Pair
