BDBM761643 2-(3-fluorophenyl)-2-(6-(4-(1- methylpiperidin-4-yl)phenyl)- 1-oxo-1,3-dihydro-2H-pyrrolo- [3,4-c]pyridin-2-yl)-N-(thiazol- 2-yl)acetamide::US12377080, Compound 6

SMILES CN1CCC(c2ccc(-c3cc4c(cn3)CN(C(C(=O)Nc3nccs3)c3cccc(F)c3)C4=O)cc2)CC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 761643   

LigandPNGBDBM761643(2-(3-fluorophenyl)-2-(6-(4-(1- methylpiperidin-4-y...)
Affinity DataIC50: 6nMAssay Description:EGFR biochemical activity measurements were carried out using the homogeneous time-resolved fluorescence (HTRF) assay (Cisbio). Inhibitors and DMSO n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM761643(2-(3-fluorophenyl)-2-(6-(4-(1- methylpiperidin-4-y...)
Affinity DataIC50: 60nMAssay Description:EGFR biochemical activity measurements were carried out using the homogeneous time-resolved fluorescence (HTRF) assay (Cisbio). Inhibitors and DMSO n...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent