BDBM762525 US12378241, Compound 1

SMILES Cn1cc(-c2ccn3c(-c4cc(CS(=O)(=O)C5CC5)nc(-c5ccc(F)cc5F)c4)cnc3c2)cn1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 762525   

LigandPNGBDBM762525(US12378241, Compound 1)
Affinity DataIC50: 2.86nMAssay Description:The IC50 value was determined using 33P isotope-labeled kinase activity test (Reaction Biology Corp) to evaluate the inhibitory ability of the compou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762525(US12378241, Compound 1)
Affinity DataIC50: 3.82nMAssay Description:The IC50 value was determined using 33P isotope-labeled kinase activity test (Reaction Biology Corp) to evaluate the inhibitory ability of the compou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent

LigandPNGBDBM762525(US12378241, Compound 1)
Affinity DataIC50: 4.55nMAssay Description:The IC50 value was determined using 33P isotope-labeled kinase activity test (Reaction Biology Corp) to evaluate the inhibitory ability of the compou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent