BDBM762527 US12378241, Compound 3

SMILES CCOC(=O)Nc1cc(-c2cnc3cc(-c4cnn(C)c4)ccn23)cc(-c2ccc(F)cc2F)n1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 762527   

TargetVascular endothelial growth factor receptor 2(Human)
Cgenetech (Suzhou,China)

US Patent
LigandPNGBDBM762527(US12378241, Compound 3)
Affinity DataIC50: 1.99nMAssay Description:The IC50 value was determined using 33P isotope-labeled kinase activity test (Reaction Biology Corp) to evaluate the inhibitory ability of the compou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent

TargetFibroblast growth factor receptor 2(Human)
Cgenetech (Suzhou,China)

US Patent
LigandPNGBDBM762527(US12378241, Compound 3)
Affinity DataIC50: 3.26nMAssay Description:The IC50 value was determined using 33P isotope-labeled kinase activity test (Reaction Biology Corp) to evaluate the inhibitory ability of the compou...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/17/2025
Entry Details
US Patent