BDBM762708 US12378251, Compound S10

SMILES CO[C@H]1Cc2ccccc2[C@H]1Nc1ncnc2c1nnn2C1CC(O)C(COS(N)(=O)=O)C1

InChI Key InChIKey=HLQPDOLGMKPDIE-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 762708   

LigandPNGBDBM762708(US12378251, Compound S10)
Affinity DataIC50: 100nMAssay Description:1. Preliminary Evaluation Experiment of Inhibiting NAE Enzyme Activity at the Molecular Level by CompoundsHomogeneous Time-Resolved Fluorescence (HTR...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/18/2025
Entry Details
Go to US Patent