BDBM762819 US20250248973, Compound 228

SMILES NS(=O)(=O)O[C@H]1C[C@@H](N/C(=N\S(=O)(=O)c2ccc(C(F)(F)F)cc2)N2C[C@@H](c3ccccc3)C(c3ccc(Cl)cc3)=N2)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 762819   

TargetIsoform 3 of Cannabinoid receptor 1(Human)
Corbus Pharmaceuticals

US Patent
LigandPNGBDBM762819(US20250248973, Compound 228)
Affinity DataIC50: 100nMAssay Description:hCB1/hCB1 b Gai Cyclic AMP (cAMP) Assays: Cells were seeded in a 384-well plate at an appropriate density from frozen cells. The cAMP assays were per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/21/2025
Entry Details
US Patent

TargetCB1 cannabinoid receptor-interacting protein 1(Human)
Corbus Pharmaceuticals

US Patent
LigandPNGBDBM762819(US20250248973, Compound 228)
Affinity DataIC50: 500nMAssay Description:hCB1/hCB1 b Gai Cyclic AMP (cAMP) Assays: Cells were seeded in a 384-well plate at an appropriate density from frozen cells. The cAMP assays were per...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/21/2025
Entry Details
US Patent