BDBM762831 (S)—N-(1-cyano-2-(2-fluoro-4-(1''-(oxetan-3-yl)-3H-spiro[isobenzofuran-1,4''-piperidin]-6-yl)phenyl)ethyl)-3-(difluoromethyl)azetidine-3-carboxamide::US20250250232, Example 15

SMILES N#C[C@H](Cc1ccc(-c2ccc3c(c2)C2(CCN(C4COC4)CC2)OC3)cc1F)NC(=O)C1(C(F)F)CNC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 762831   

TargetDipeptidyl peptidase 1(Human)TBA
LigandPNGBDBM762831((S)—N-(1-cyano-2-(2-fluoro-4-(1'-(oxetan-3-yl)-3H-...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
TBA
Entry Details
US Patent