BDBM762856 Single enantiomers of N-(1-cyano-2-(5-(4-cyanophenyl)-3-fluoropyridin-2-yl)ethyl)-3-methoxy-1-methylazetidine-3-carboxamide (enantiomers 1 and 2)::US20250250232, Example 44

SMILES COC1(C(=O)NC(C#N)Cc2ncc(-c3ccc(C#N)cc3)cc2F)CN(C)C1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 762856   

TargetDipeptidyl peptidase 1(Human)
Chiesi Farmaceutici

US Patent
LigandPNGBDBM762856(Single enantiomers of N-(1-cyano-2-(5-(4-cyanophen...)
Affinity DataIC50: 55nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/21/2025
Entry Details
US Patent