BDBM762861 (S)-N-(1-cyano-2-(2-fluoro-4-(1- methyl-2-oxoindolin-6- yl)phenyl)ethyl)-3- methoxyazetidine-3- carboxamide::US20250250232, Example 49

SMILES COC1(C(=O)N[C@H](C#N)Cc2ccc(-c3ccc4c(c3)N(C)C(=O)C4)cc2F)CNC1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 762861   

TargetDipeptidyl peptidase 1(Human)
Chiesi Farmaceutici

US Patent
LigandPNGBDBM762861((S)-N-(1-cyano-2-(2-fluoro-4-(1- methyl-2-oxoindol...)
Affinity DataIC50: 10nMAssay Description:Human DPP1 enzyme activity was determined by measuring release of the fluorophore aminomethyl coumarin (AMC) following enzymatic cleavage of the dipe...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/21/2025
Entry Details
US Patent