BDBM763808 5-[4-({4''-fluoro-[1,1-biphenyl]- 2-yl}amino)phenyl]-1,3,4- thiadiazol-2-amine::US12384772, Compound 505

SMILES Nc1nnc(-c2ccc(Nc3ccccc3-c3ccc(F)cc3)cc2)s1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 763808   

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763808(5-[4-({4'-fluoro-[1,1-biphenyl]- 2-yl}amino)phenyl...)
Affinity DataKi:  1.52E+3nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763808(5-[4-({4'-fluoro-[1,1-biphenyl]- 2-yl}amino)phenyl...)
Affinity DataKi:  1.81E+3nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent