BDBM763809 5-(4-{[2-(3,4- dimethoxyphenyl)phenyl]amino} phenyl)-1,3,4-thiadiazol-2- amine::US12384772, Compound 561

SMILES COc1ccc(-c2ccccc2Nc2ccc(-c3nnc(N)s3)cc2)cc1OC

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 763809   

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763809(5-(4-{[2-(3,4- dimethoxyphenyl)phenyl]amino} pheny...)
Affinity DataKi:  420nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763809(5-(4-{[2-(3,4- dimethoxyphenyl)phenyl]amino} pheny...)
Affinity DataKi:  1.09E+3nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent