BDBM763818 5-[4-({2-[4-(propan-2- yloxy)phenyl]phenyl}amino)phe- nyl]-1,3,4-thiadiazol-2-amine::US12384772, Compound 1296

SMILES CC(C)Oc1ccc(-c2ccccc2Nc2ccc(-c3nnc(N)s3)cc2)cc1

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 763818   

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763818(5-[4-({2-[4-(propan-2- yloxy)phenyl]phenyl}amino)p...)
Affinity DataKi:  1.51E+3nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763818(5-[4-({2-[4-(propan-2- yloxy)phenyl]phenyl}amino)p...)
Affinity DataKi:  3.27E+3nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent