BDBM763820 3'',4''-dimethoxy-N-[4-(4-methyl- 4H-1,2,4-triazol-3-yl)phenyl]- [1,1''-biphenyl]-2-amine::US12384772, Compound 854

SMILES COc1ccc(-c2ccccc2Nc2ccc(-c3nncn3C)cc2)cc1OC

InChI Key

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 763820   

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763820(3',4'-dimethoxy-N-[4-(4-methyl- 4H-1,2,4-triazol-3...)
Affinity DataKi:  440nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent

TargetGlutaminyl-peptide cyclotransferase(Human)
Vivoryon Therapeutics

US Patent
LigandPNGBDBM763820(3',4'-dimethoxy-N-[4-(4-methyl- 4H-1,2,4-triazol-3...)
Affinity DataKi:  1.48E+3nMAssay Description:10 mM compound stock solutions were prepared in DMSO. For IC50 determination compound stocks were serially diluted (1:3) in DMSO.All measurements wer...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
11/24/2025
Entry Details
US Patent